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微波辅助有机化学对药物发现的影响。

The impact of microwave-assisted organic chemistry on drug discovery.

作者信息

Wathey Bernard, Tierney Jason, Lidström Pelle, Westman Jacob

机构信息

BioFocus, 130, Abbott Drive, Sittingbourne Research Centre, Sittingbourne, Kent, UK ME9 8AZ.

出版信息

Drug Discov Today. 2002 Mar 15;7(6):373-80. doi: 10.1016/s1359-6446(02)02178-5.

DOI:10.1016/s1359-6446(02)02178-5
PMID:11893546
Abstract

Microwave-assisted organic synthesis (MAOS) is rapidly becoming recognized as a valuable tool for easing some of the bottlenecks in the drug discovery process. This article outlines the basic principles behind the technology and summarizes the areas in which microwave technology has made an impact, to date.

摘要

微波辅助有机合成（MAOS）正迅速成为一种有价值的工具，用于缓解药物研发过程中的一些瓶颈。本文概述了该技术背后的基本原理，并总结了迄今为止微波技术产生影响的领域。

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