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Facile one-pot synthesis of aromatic and heteroaromatic sulfonamides.

作者信息

Pandya Rina, Murashima Takashi, Tedeschi Livio, Barrett Anthony G M

机构信息

Department of Chemistry, Imperial College London, London SW7 2AZ, England.

出版信息

J Org Chem. 2003 Oct 17;68(21):8274-6. doi: 10.1021/jo034643j.

DOI:10.1021/jo034643j
PMID:14535819
Abstract

A series of arene and heteroarene sulfonamides were prepared in one vessel from aryl and heteroaryl bromides via conversion into the corresponding Grignard reagents using either magnesium or isopropylmagnesium chloride and subsequent reaction with sulfur dioxide, sulfuryl chloride, and an amine.

摘要

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