一种高效的融合吲哚啉的方法，通过铜（I）催化磺酰叠氮与 2-乙炔基芳基亚甲基环丙烷的反应。
An efficient approach to fused indolines via a copper(I)-catalyzed reaction of sulfonyl azide with 2-ethynylaryl methylenecyclopropane.
机构信息
Department of Chemistry, Fudan University, 220 Handan Road, Shanghai 200433, China.
出版信息
Org Lett. 2011 Jun 17;13(12):3190-3. doi: 10.1021/ol2011067. Epub 2011 May 23.
PMID:21604754
Abstract
A cascade reaction of 2-ethynylaryl methylenecyclopropane with sulfonyl azide catalyzed by copper(I) iodide under mild conditions is described, which provides a novel and efficient route for the generation of fused indolines.
摘要
碘化亚铜催化温和条件下 2-乙炔基芳基亚甲基环丙烷与磺酰叠氮的级联反应，为构建稠合吲哚啉提供了一种新颖、高效的方法。
Zotero 插件