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1
Towards an in vitro model of Plasmodium hypnozoites suitable for drug discovery.
PLoS One. 2011 Mar 31;6(3):e18162. doi: 10.1371/journal.pone.0018162.
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A research agenda for malaria eradication: drugs.
PLoS Med. 2011 Jan 25;8(1):e1000402. doi: 10.1371/journal.pmed.1000402.
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Falcipain inhibitors: optimization studies of the 2-pyrimidinecarbonitrile lead series.
J Med Chem. 2010 Aug 26;53(16):6129-52. doi: 10.1021/jm100556b.
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Visualisation and quantitative analysis of the rodent malaria liver stage by real time imaging.
PLoS One. 2009 Nov 18;4(11):e7881. doi: 10.1371/journal.pone.0007881.
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New medicines to improve control and contribute to the eradication of malaria.
Nat Rev Drug Discov. 2009 Nov;8(11):879-91. doi: 10.1038/nrd2972. Epub 2009 Oct 16.
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Hybrid drugs for malaria.
Curr Pharm Des. 2009;15(25):2970-85. doi: 10.2174/138161209789058183.
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Artemisinin-dipeptidyl vinyl sulfone hybrid molecules: design, synthesis and preliminary SAR for antiplasmodial activity and falcipain-2 inhibition.
Bioorg Med Chem Lett. 2009 Jun 15;19(12):3229-32. doi: 10.1016/j.bmcl.2009.04.100. Epub 2009 May 3.

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