通过硫叶立德和 N-(邻氯甲基)芳酰胺的高效级联反应合成吲哚。
Synthesis of indoles through highly efficient cascade reactions of sulfur ylides and N-(ortho-chloromethyl)aryl amides.
机构信息
Key Laboratory of Pesticide & Chemical Biology, Ministry of Education, College of Chemistry, Central China Normal University, Wuhan, Hubei 430079, China.
出版信息
Angew Chem Int Ed Engl. 2012 Sep 3;51(36):9137-40. doi: 10.1002/anie.201203657. Epub 2012 Aug 6.
PMID:22888071
Abstract
Batting the ylides: A simple procedure carried out under mild conditions allows the direct and efficient synthesis of structurally diverse indoles. This approach involves a cascade reaction of sulfur ylides and N-(ortho-chloromethyl)aryl amides.
摘要
叶立德反应
在温和条件下进行的简单操作可实现结构多样吲哚的直接、高效合成。该方法涉及硫叶立德与 N-（邻氯甲基）芳酰胺的级联反应。
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