碘催化吲哚与亚硫酸钠的区域选择性 2-磺酰化反应。
Iodine-catalyzed regioselective 2-sulfonylation of indoles with sodium sulfinates.
机构信息
Key Laboratory of Environmentally Friendly Chemistry and Application of Ministry of Education, College of Chemistry, Xiangtan University , Xiangtan 411105, China.
出版信息
Org Lett. 2014 Jan 3;16(1):50-3. doi: 10.1021/ol402987u. Epub 2013 Dec 11.
PMID:24328422
Abstract
Iodine-catalyzed selective 2-arylsulfonyl indole formation from indoles and sodium sulfinates is disclosed. Various substituted 2-arylsulfonyl indoles were obtained in one pot in the absence of metal catalyst at room temperature under air.
摘要
碘催化吲哚与亚磺酸钠的选择性 2-芳磺酰吲哚形成反应被揭示。在室温下、空气中、无需金属催化剂的条件下，一锅法可得到各种取代的 2-芳磺酰吲哚。
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