Key Laboratory for Functional Material, Educational Department of Liaoning Province, University of Science and Technology Liaoning, Anshan, 114051, P. R. China.
Org Biomol Chem. 2014 Mar 21;12(11):1721-4. doi: 10.1039/c3ob42171f.
An efficient Cu-catalyzed decarboxylative C3-acylation of free (N-H) indoles using α-oxocarboxylic acids as acylating agents has been developed. This method was compatible with a variety of functional groups and provided an attractive alternative access to 3-acylindoles in moderate to high yields.
一种高效的 Cu 催化的脱羧 C3-酰化游离（N-H）吲哚的方法已经被开发出来，该方法使用α-氧代羧酸作为酰化试剂。该方法与多种官能团兼容，并提供了一种有吸引力的替代方法，以中等到高产率得到 3-酰基吲哚。
