磷酸泰地唑胺（西沃沙星）：一种用于治疗急性细菌性皮肤及皮肤结构感染的第二代恶唑烷酮类药物。
Tedizolid phosphate (sivextro): a second-generation oxazolidinone to treat acute bacterial skin and skin structure infections.
作者信息
Wong Elaine, Rab Saba
出版信息
P T. 2014 Aug;39(8):555-79.
Abstract
Tedizolid phosphate: a second-generation oxazolidinone for acute bacterial skin and skin structure infections.
摘要
磷酸泰地唑胺
一种用于治疗急性细菌性皮肤及皮肤结构感染的第二代恶唑烷酮类药物。
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本文引用的文献
1
Tedizolid for 6 days versus linezolid for 10 days for acute bacterial skin and skin-structure infections (ESTABLISH-2): a randomised, double-blind, phase 3, non-inferiority trial.替考拉宁治疗 6 天与利奈唑胺治疗 10 天治疗急性细菌性皮肤和皮肤结构感染（ESTABLISH-2）：一项随机、双盲、III 期、非劣效性试验。
Lancet Infect Dis. 2014 Aug;14(8):696-705. doi: 10.1016/S1473-3099(14)70737-6. Epub 2014 Jun 5.
2
FDA guidance for ABSSSI trials: implications for conducting and interpreting clinical trials.FDA 指导意见下的 ABSSSI 临床试验：对临床试验开展和解读的影响。
Clin Infect Dis. 2014 Jan;58 Suppl 1:S4-9. doi: 10.1093/cid/cit612.
3
In vitro, in vivo, and clinical studies of tedizolid to assess the potential for peripheral or central monoamine oxidase interactions.体外、体内和临床研究替加环素，以评估潜在的外周或中枢单胺氧化酶相互作用。
Antimicrob Agents Chemother. 2013 Jul;57(7):3060-6. doi: 10.1128/AAC.00431-13. Epub 2013 Apr 22.
4
Tedizolid phosphate vs linezolid for treatment of acute bacterial skin and skin structure infections: the ESTABLISH-1 randomized trial.磷酸替加环素与利奈唑胺治疗急性细菌性皮肤和皮肤结构感染：ESTABLISH-1 随机试验。
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Comparative pharmacodynamics of the new oxazolidinone tedizolid phosphate and linezolid in a neutropenic murine Staphylococcus aureus pneumonia model.新恶唑烷酮类药物替加环素磷酸盐与利奈唑胺在中性粒细胞减少的金黄色葡萄球菌肺炎小鼠模型中的比较药效学研究。
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Activity of tedizolid phosphate (TR-701) in murine models of infection with penicillin-resistant and penicillin-sensitive Streptococcus pneumoniae.磷酸泰地唑利（TR-701）在耐青霉素和青霉素敏感肺炎链球菌感染的小鼠模型中的活性。
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Comparative efficacies of human simulated exposures of tedizolid and linezolid against Staphylococcus aureus in the murine thigh infection model.替加环素与利奈唑胺在小鼠大腿感染模型中抗金黄色葡萄球菌的人体模拟暴露比较疗效。
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Skin and soft tissue concentrations of tedizolid (formerly torezolid), a novel oxazolidinone, following a single oral dose in healthy volunteers.健康志愿者单次口服替加环素（原称替唑肟）后的皮肤和软组织浓度。
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