2-碘异吲哚酮：用于合成氮杂环的多功能中间体。
2-Iodoisatogens: versatile intermediates for the synthesis of nitrogen heterocycles.
作者信息
Maduli Elvis J M, Edeson Steven J, Swanson Stephen, Procopiou Panayiotis A, Harrity Joseph P A
机构信息
Department of Chemistry, University of Sheffield , Sheffield S3 7HF, U.K.
出版信息
Org Lett. 2015 Jan 16;17(2):390-2. doi: 10.1021/ol503487f. Epub 2014 Dec 23.
PMID:25536211
Abstract
A Cu-promoted cyclization of 2-nitrophenyl iodoacetylenes provides a direct route to a range of 2-iodoisatogens. These compounds represent useful intermediates for the late-stage elaboration of the C-I bond to furnish isatins and a range of alternative heterocyclic products.
摘要
铜促进的2-硝基苯基碘乙炔环化反应提供了一条直接合成一系列2-碘异吲哚酮的途径。这些化合物是后期将碳-碘键转化为异吲哚酮及一系列其他杂环产物的有用中间体。
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