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Activity of esterase in the hydrolysis of 3',5'-diesters of 5-fluoro-2'-deoxyuridine in relation to the structure of the diester prodrugs.

作者信息

Kawaguchi T, Suzuki Y, Nakahara Y, Nambu N, Nagai T

出版信息

Chem Pharm Bull (Tokyo). 1985 Jan;33(1):301-7. doi: 10.1248/cpb.33.301.

DOI:10.1248/cpb.33.301
PMID:3159490
Abstract
摘要

相似文献

1
Activity of esterase in the hydrolysis of 3',5'-diesters of 5-fluoro-2'-deoxyuridine in relation to the structure of the diester prodrugs.酯酶在5-氟-2'-脱氧尿苷3',5'-二酯水解中的活性与二酯前药结构的关系
Chem Pharm Bull (Tokyo). 1985 Jan;33(1):301-7. doi: 10.1248/cpb.33.301.
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J Pharm Sci. 1988 Oct;77(10):855-60. doi: 10.1002/jps.2600771009.

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Nonenzymatic and enzymatic hydrolysis of 5-fluoro-2'-deoxyuridine (FUdR) esters.5-氟-2'-脱氧尿苷(FUdR)酯的非酶促水解和酶促水解
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Chemical and enzymatic degradation of ganciclovir prodrugs: enhanced stability of the diadamantoate prodrug under acid conditions.
Pharm Res. 1991 Nov;8(11):1418-23. doi: 10.1023/a:1015809408908.