醋酸碘苯介导的分子内氧化碳氮偶联及脱对甲苯磺酰基芳构化反应：一种合成吲哚并[2,3 -]喹啉的方法
PhI(OAc)-mediated intramolecular oxidative C-N coupling and detosylative aromatization: an access to indolo[2,3-]quinolines.
作者信息
Wang Quan-Bing, Tang Shi, Wang Ying-Jie, Yuan Yue, Chen Tieqiao, Jia Ai-Qun
机构信息
School of Life and Pharmaceutical Sciences, Key Laboratory of Tropical Biological Resources of Ministry of Education, Hainan University Haikou 570228 China
出版信息
RSC Adv. 2021 May 10;11(28):17206-17211. doi: 10.1039/d1ra01894a. eCollection 2021 May 6.
Abstract
A PIDA mediated intramolecular oxidative C-N coupling and subsequent detosylative aromatization to afford indolo[2,3-]quinoline derivatives has been developed. This tandem reaction provided an efficient method for the synthesis of valuable indolo[2,3-]quinoline derivatives.
摘要
已开发出一种由PIDA介导的分子内氧化C-N偶联及随后的脱对甲苯磺酰基芳构化反应，以得到吲哚并[2,3 -]喹啉衍生物。这种串联反应为合成有价值的吲哚并[2,3 -]喹啉衍生物提供了一种有效方法。
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