吡咯菌素类似物。十二。某些吡唑羧酸的合成与生物活性。
Pyrrolnitrin analogues. XII. Synthesis and biological activity of some pyrazole carboxylic acids.
作者信息
Palazzino G, Melani F, Cecchi L, Filacchioni G
出版信息
Farmaco Sci. 1986 Jul;41(7):566-76.
PMID:3743749
Abstract
Some 1,5-diaryl-, 1-aryl-5-(2-nitrobenzyl)-3-methylpyraloze-4-carboxylic acids and some of their 4-morpholino- and 4-N-methylpiperazino amides are prepared and tested as antibacterial agents. None of the tested compounds shows any noteworthy antimicrobial activity. The results are discussed and compared with the previously published results for other similarly structured compounds.
摘要
制备了一些1,5 - 二芳基 - 、1 - 芳基 - 5 - (2 - 硝基苄基) - 3 - 甲基吡唑 - 4 - 羧酸及其一些4 - 吗啉代和4 - N - 甲基哌嗪酰胺，并作为抗菌剂进行了测试。所测试的化合物均未显示出任何值得注意的抗菌活性。对结果进行了讨论，并与先前发表的其他结构类似化合物的结果进行了比较。
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