Irreversible enzyme inhibitors. 143. Active-site-directed irreversible inhibitors of dihydrofolic reductase derived from 5-(p-aminophenoxypropyl)-2,4-diamino-6-methylpyrimidine with a terminal sulfonyl fluoride.
作者信息
Baker B R, Meyer R B
出版信息
J Med Chem. 1969 Jan;12(1):108-11. doi: 10.1021/jm00301a028.