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[35S]t-butylbicyclophosphorothionate binds with high affinity to brain-specific sites coupled to gamma-aminobutyric acid-A and ion recognition sites.

作者信息

Squires R F, Casida J E, Richardson M, Saederup E

出版信息

Mol Pharmacol. 1983 Mar;23(2):326-36.

PMID:6300642
Abstract
摘要

相似文献

1
[35S]t-butylbicyclophosphorothionate binds with high affinity to brain-specific sites coupled to gamma-aminobutyric acid-A and ion recognition sites.[35S]叔丁基双环硫代磷酸酯与与γ-氨基丁酸-A和离子识别位点偶联的脑特异性位点具有高亲和力结合。
Mol Pharmacol. 1983 Mar;23(2):326-36.
2
t-[3H]butylbicycloorthobenzoate: new radioligand probe for the gamma-aminobutyric acid-regulated chloride ionophore.t-[3H]丁基双环原苯甲酸酯：一种用于γ-氨基丁酸调节氯离子通道的新型放射性配体探针。
J Neurochem. 1985 Sep;45(3):798-804. doi: 10.1111/j.1471-4159.1985.tb04063.x.
3
Solubilization of convulsant/barbiturate binding activity on the gamma-aminobutyric acid/benzodiazepine receptor complex.
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4
Dependence on gamma-aminobutyric acid of pyrethroid and 4'-chlorodiazepam modulation of the binding of t-[35S]butylbicyclophosphorothionate in piscine brain.
Neuropharmacology. 1990 Jul;29(7):641-8. doi: 10.1016/0028-3908(90)90025-m.
5
Effect of benzodiazepine binding site ligands on [35S] t-butylbicyclophosphorothionate ([35S]TBPS) binding to rat brain: an autoradiographic study.苯二氮䓬结合位点配体对[35S]叔丁基双环磷硫代酸盐（[35S]TBPS）与大鼠脑结合的影响：一项放射自显影研究。
Adv Biochem Psychopharmacol. 1986;41:227-38.
6
Alkyl-substituted gamma-butyrolactones inhibit [35S]TBPS binding to a GABA linked chloride ionophore.
Eur J Pharmacol. 1984 Oct 1;105(1-2):195-6. doi: 10.1016/0014-2999(84)90669-1.
7
Similar properties of [35S]t-butylbicyclophosphorothionate receptor and coupled components of the GABA receptor-ionophore complex in brains of human, cow, rat, chicken and fish.
Life Sci. 1984 Oct 22;35(17):1755-62. doi: 10.1016/0024-3205(84)90272-8.
8
RO5-4864 inhibits the binding of [35S]t-butylbicyclophosphorothionate to rat brain membranes.
Life Sci. 1984 Feb 13;34(7):631-8. doi: 10.1016/0024-3205(84)90226-1.
9
[35S]tert.-butylbicyclophosphorothionate and avermectin bind to different sites associated with the gamma- aminobutyric acid-benzodiazepine receptor complex.[35S]叔丁基双环硫代磷酸酯和阿维菌素与γ-氨基丁酸-苯二氮䓬受体复合物相关的不同位点结合。
Neurosci Lett. 1984 Sep 7;50(1-3):273-7. doi: 10.1016/0304-3940(84)90498-1.
10
Barbiturate recognition site on the GABA/benzodiazepine receptor complex is distinct from the picrotoxinin/TBPS recognition site.
Eur J Pharmacol. 1984 Nov 13;106(2):441-7. doi: 10.1016/0014-2999(84)90737-4.

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