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一株甲硝唑耐药性阴道毛滴虫及其对Go 10213的敏感性

A metronidazole-resistant strain of Trichomonas vaginalis and its sensitivity to Go 10213.

作者信息

Ray D K, Tendulkar J S, Shrivastava V B, Datta A K, Nagarajan K

出版信息

J Antimicrob Chemother. 1984 Oct;14(4):423-6. doi: 10.1093/jac/14.4.423.

DOI:10.1093/jac/14.4.423
PMID:6334072
Abstract

In the present study the comparative in-vitro and in-vivo efficacy of Go 10213 was compared with those of metronidazole, secnidazole, tinidazole, ornidazole and nimorazole against a metronidazole-resistant strain of T. vaginalis. Go 10213 was found to be superior in activity. It appears more promising than the drugs mentioned above on the basis of the evidence presented.

摘要

在本研究中,将Go 10213与甲硝唑、塞克硝唑、替硝唑、奥硝唑和尼莫唑针对一株甲硝唑耐药的阴道毛滴虫进行了体外和体内疗效比较。结果发现Go 10213活性更强。根据所提供的证据,它似乎比上述药物更具前景。

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引用本文的文献

1
Secnidazole for Trichomoniasis in Women and Men.硝呋太尔用于治疗女性和男性滴虫病。
Sex Med Rev. 2022 Apr;10(2):255-262. doi: 10.1016/j.sxmr.2021.12.004. Epub 2022 Feb 10.
2
Secnidazole. A review of its antimicrobial activity, pharmacokinetic properties and therapeutic use in the management of protozoal infections and bacterial vaginosis.塞克硝唑。对其抗菌活性、药代动力学特性以及在原生动物感染和细菌性阴道病治疗中的应用综述。
Drugs. 1996 Apr;51(4):621-38. doi: 10.2165/00003495-199651040-00007.
3
Antibacterial activity of GO 10213, a nitroimidazole derivative.
硝基咪唑衍生物GO 10213的抗菌活性
Antimicrob Agents Chemother. 1986 May;29(5):953-4. doi: 10.1128/AAC.29.5.953.
4
Anti-Trichomonas vaginalis monoclonal antibodies inducing complement-dependent cytotoxicity.诱导补体依赖性细胞毒性的抗阴道毛滴虫单克隆抗体。
Immunology. 1988 Jan;63(1):63-9.