亚胺培南对普通变形杆菌β-内酰胺酶抑制作用的动力学研究
Kinetic studies on the inhibition of Proteus vulgaris beta-lactamase by imipenem.
作者信息
Hashizume T, Yamaguchi A, Hirata T, Sawai T
出版信息
Antimicrob Agents Chemother. 1984 Jan;25(1):149-51. doi: 10.1128/AAC.25.1.149.
Abstract
Imipenem was found to inhibit Proteus vulgaris beta-lactamase in a progressive manner. Kinetic experiments confirmed that the inactivated enzyme was not completely recovered after intact imipenem had been exhausted.
摘要
发现亚胺培南能以渐进方式抑制普通变形杆菌β-内酰胺酶。动力学实验证实，当完整的亚胺培南耗尽后，失活的酶不能完全恢复。
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