英普咪定（SK&F 92676）对大鼠离体全胃起部分激动剂的作用。
Impromidine (SK & F 92676) acts as a partial agonist on the isolated whole stomach of the rat.
作者信息
Parsons M, Sykes C
出版信息
Br J Pharmacol. 1980 May;69(1):6-7. doi: 10.1111/j.1476-5381.1980.tb10874.x.
Abstract
The present secretory studies on the isolated stomach of the rat provide evidence that impromidine acts as a partial agonist at the histamine H2-receptors. It was found to be 100 times more potent than histamine but with a maximal response only 50% that obtained with histamine.
摘要
目前对大鼠离体胃的分泌研究提供了证据，表明英普咪定在组胺H2受体上作为部分激动剂起作用。发现它的效力比组胺高100倍，但最大反应仅为组胺的50%。
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Impromidine (SK & F 92676) acts as a partial agonist on the isolated whole stomach of the rat.英普咪定（SK&F 92676）对大鼠离体全胃起部分激动剂的作用。
Br J Pharmacol. 1980 May;69(1):6-7. doi: 10.1111/j.1476-5381.1980.tb10874.x.
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本文引用的文献
1
Impromidine (SK&F 92676) is a very potent and specific agonist for histamine H2 receptors.英普咪定（SK&F 92676）是一种效力很强且特异性很高的组胺H2受体激动剂。
Nature. 1978 Nov 23;276(5686):403-5. doi: 10.1038/276403a0.
2
A quantitative study of metiamide, a histamine H2-antagonist, on the isolated whole rat stomach.组胺H2拮抗剂甲硫米特对离体大鼠全胃作用的定量研究。
J Physiol. 1976 Jun;258(2):453-65. doi: 10.1113/jphysiol.1976.sp011430.
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