Design of more potent and selective antagonists of the antidiuretic responses to arginine-vasopressin devoid of antidiuretic agonism.

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超能文献

作者信息

Manning M, Klis W A, Olma A, Seto J, Sawyer W H

出版信息

J Med Chem. 1982 Apr;25(4):414-9. doi: 10.1021/jm00346a016.

DOI:10.1021/jm00346a016

PMID:7069720

Abstract

摘要

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Stimulation of vasopressin release in the ventral septum of the rat brain suppresses prostaglandin E1 fever.刺激大鼠脑腹侧隔区中血管加压素的释放可抑制前列腺素E1引起的发热。

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