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Platelet aggregation inhibitors. IX. Chemical transformation of adenosine into 2-thioadenosine derivatives.

作者信息

Kikugawa K, Suehiro H, Yanase R, Aoki A

出版信息

Chem Pharm Bull (Tokyo). 1977 Aug;25(8):1959-69. doi: 10.1248/cpb.25.1959.

DOI:10.1248/cpb.25.1959
PMID:922979
Abstract
摘要

相似文献

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Chem Pharm Bull (Tokyo). 1977 Aug;25(8):1959-69. doi: 10.1248/cpb.25.1959.
2
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New inhibitors of platelet aggregation. 5'-Phosphate, 5'-phosphorothioate, and 5'-O-sulfamoyl derivatives of 2-substituted adenosine analogues.血小板聚集的新型抑制剂。2-取代腺苷类似物的5'-磷酸酯、5'-硫代磷酸酯和5'-O-氨磺酰衍生物。
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5'-Methylthioadenosine and 2',5'-dideoxyadenosine blockade of the inhibitory effects of adenosine on ADP-induced platelet aggregation by different mechanisms.5'-甲硫基腺苷和2',5'-二脱氧腺苷通过不同机制阻断腺苷对二磷酸腺苷诱导的血小板聚集的抑制作用。
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J Med Chem. 1993 Nov 26;36(24):3937-46. doi: 10.1021/jm00076a023.
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Specific but noncompetitive inhibition by 2-alkylthio analogues of adenosine 5'-monophosphate and adenosine 5'-triphosphate of human platelet aggregation induced by adenosine 5'-diphosphate.5'-二磷酸腺苷诱导的人血小板聚集受到5'-单磷酸腺苷和5'-三磷酸腺苷的2-烷硫基类似物的特异性而非竞争性抑制。
Br J Pharmacol. 1982 Feb;75(2):397-400. doi: 10.1111/j.1476-5381.1982.tb08800.x.
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