（Z）-二甲基氨基-1-（4-溴苯基）-1-（3-吡啶基）丙烯（h 102/09），一种新型的神经元5-羟色胺摄取选择性抑制剂。 - Suppr

Suppr

超能文献

(Z)-dimethylamino-1-(4-bromophenyl)-1-(3-pyridyl) propene (h 102/09), a new selective inhibitor of the neuronal 5-hydroxytryptamine uptake.

作者信息

Ross S B, Ogren S O, Renyi A L

出版信息

Acta Pharmacol Toxicol (Copenh). 1976 Aug;39(2):152-66. doi: 10.1111/j.1600-0773.1976.tb03166.x.

DOI:10.1111/j.1600-0773.1976.tb03166.x

PMID:947293

Abstract

摘要

相似文献

(Z)-dimethylamino-1-(4-bromophenyl)-1-(3-pyridyl) propene (h 102/09), a new selective inhibitor of the neuronal 5-hydroxytryptamine uptake.（Z）-二甲基氨基-1-（4-溴苯基）-1-（3-吡啶基）丙烯（h 102/09），一种新型的神经元5-羟色胺摄取选择性抑制剂。

Acta Pharmacol Toxicol (Copenh). 1976 Aug;39(2):152-66. doi: 10.1111/j.1600-0773.1976.tb03166.x.

Inhibition of the neuronal uptake of 5-hydroxytryptamine and noradrenaline in rat brain by (Z)- and (E)-3-(4-bromophenyl)-N,N-dimethyl-3-(3-pyridyl) allylamines and their secondary analogues.（Z）-和（E）-3-（4-溴苯基）-N，N-二甲基-3-（3-吡啶基）烯丙胺及其二级类似物对大鼠脑内5-羟色胺和去甲肾上腺素神经元摄取的抑制作用

Neuropharmacology. 1977 Jan;16(1):57-63. doi: 10.1016/0028-3908(77)90048-x.

Effect of etoperidone on the depletion of brain 5-hydroxytryptamine and catecholamines induced respectively by p-chloromethamphetamine and 6-hydroxydopamine in rats.依托哌酮对大鼠中由对氯甲基苯丙胺和6-羟基多巴胺分别诱导的脑5-羟色胺和儿茶酚胺耗竭的影响。

Pharmacol Res Commun. 1979 Feb;11(2):169-77. doi: 10.1016/s0031-6989(79)80070-3.

Effect of butriptyline on the brain uptake mechanisms for noradrenaline and 5-hydroxytryptamine.布替林对去甲肾上腺素和5-羟色胺脑摄取机制的影响。

J Pharm Pharmacol. 1974 Oct;26(10):778-8. doi: 10.1111/j.2042-7158.1974.tb09173.x.

Substituted amphetamine derivatives. I. Effect on uptake and release of biogenic monoamines and on monoamine oxidase in the mouse brain.取代苯丙胺衍生物。I. 对小鼠脑中生物源性单胺的摄取和释放以及单胺氧化酶的影响。

Acta Pharmacol Toxicol (Copenh). 1977 Oct;41(4):337-52. doi: 10.1111/j.1600-0773.1977.tb02673.x.

Dopamine but not norepinephrine or serotonin uptake inhibitors protect mice against neurotoxicity of MPTP.

Eur J Pharmacol. 1985 Oct 8;116(1-2):179-81. doi: 10.1016/0014-2999(85)90201-8.

Differences between the effects of acute and long-term treatment with desmethylimipramine on reserpine-induced release of amines from rat brain.去甲丙咪嗪急性治疗与长期治疗对利血平诱导的大鼠脑内胺类释放的影响差异。

Biochem Pharmacol. 1975 Jul 15;24(13-14):1321-5. doi: 10.1016/0006-2952(75)90346-9.

Antagonism of the acute and long-term biochemical effects of 4-chloroamphetamine on the 5-HT neurones in the rat brain by inhibitors of the 5-hydroxytryptamine uptake.5-羟色胺摄取抑制剂对4-氯苯丙胺对大鼠脑内5-羟色胺神经元的急性和长期生化作用的拮抗作用

Acta Pharmacol Toxicol (Copenh). 1976;39(4):456-76. doi: 10.1111/j.1600-0773.1976.tb03197.x.

Efflux of 5-hydroxytryptamine from synaptosomes of rat cerebral cortex.5-羟色胺从大鼠大脑皮质突触体的流出。

Acta Physiol Scand. 1977 Jan;99(1):27-36. doi: 10.1111/j.1748-1716.1977.tb10348.x.

Effects of Org 6582, chlorimipramine and desmethylimipramine on the depletion of biogenic amines from the rat brain in vivo.Org 6582、氯米帕明和去甲氯米帕明对大鼠脑内生物胺在体耗竭的影响。

Biochem Pharmacol. 1977 Jun 1;26(11):1083-4. doi: 10.1016/0006-2952(77)90248-9.

引用本文的文献

Prophylactic treatment with the tricyclic antidepressant desipramine prevents development of paclitaxel-induced neuropathic pain through activation of endogenous analgesic systems.使用三环类抗抑郁药地昔帕明进行预防性治疗可通过激活内源性镇痛系统来预防紫杉醇诱导的神经性疼痛的发生。

Pharmacol Res. 2016 Dec;114:75-89. doi: 10.1016/j.phrs.2016.10.007. Epub 2016 Oct 20.

In vivo electrochemical measurements of serotonin clearance in rat striatum: effects of neonatal 6-hydroxydopamine-induced serotonin hyperinnervation and serotonin uptake inhibitors.大鼠纹状体中血清素清除率的体内电化学测量：新生期6-羟基多巴胺诱导的血清素超神经支配和血清素摄取抑制剂的影响

J Neural Transm (Vienna). 1997;104(4-5):379-97. doi: 10.1007/BF01277658.

Effects of monoamine uptake inhibitors given early postnatally on monoamines in the brain stem, caudate/putamen and cortex, and on dopamine D1 and D2 receptors in the caudate/putamen.

J Neural Transm Gen Sect. 1995;102(2):139-48. doi: 10.1007/BF01276509.

Antidepressant drugs and ethanol: behavioral and pharmacokinetic interactions in mice.抗抑郁药物与乙醇：小鼠的行为及药代动力学相互作用

J Neural Transm. 1980;48(4):223-40. doi: 10.1007/BF01250658.

Further evidence for an inhibitory role of central 5-HT in male rat sexual behavior.中枢5-羟色胺对雄性大鼠性行为具有抑制作用的进一步证据。

Psychopharmacology (Berl). 1980;68(3):217-20. doi: 10.1007/BF00428106.

Inhibition of 5-hydroxytryptamine uptake in human platelets by antidepressant agents in vivo.

Psychopharmacology (Berl). 1980 Jan;67(1):1-7. doi: 10.1007/BF00427588.

Antagonism of fenfluramine-induced hyperthermia in rats by some, but not all, selective inhibitors of 5-hydroxytryptamine uptake.某些（但并非全部）5-羟色胺摄取选择性抑制剂对大鼠芬氟拉明诱导的体温过高具有拮抗作用。

Br J Pharmacol. 1984 Apr;81(4):651-7. doi: 10.1111/j.1476-5381.1984.tb16131.x.

Effects of LM 5008, a selective inhibitor of 5-hydroxytryptamine uptake, on blood pressure and responses to sympathomimetic amines.5-羟色胺摄取选择性抑制剂LM 5008对血压及对拟交感胺反应的影响。

Br J Pharmacol. 1983 Aug;79(4):915-22. doi: 10.1111/j.1476-5381.1983.tb10536.x.

Chronic treatment with antidepressants: protentiation of clonidine-induced aggression in mice via noradrenergic mechanism.抗抑郁药的长期治疗：通过去甲肾上腺素能机制增强可乐定诱导的小鼠攻击行为。

J Neural Transm. 1981;52(3):189-97. doi: 10.1007/BF01249603.

Effects of zimelidine and desipramine on serotonin and noradrenaline uptake mechanisms in relation to plasma concentrations and to therapeutic effects during treatment of depression.齐美利定和地昔帕明对5-羟色胺和去甲肾上腺素摄取机制的影响与抑郁症治疗期间的血浆浓度及治疗效果的关系。

Psychopharmacology (Berl). 1981;74(4):297-305. doi: 10.1007/BF00432735.

文献AI研究员

20分钟写一篇综述，助力文献阅读效率提升50倍。

立即体验

用中文搜PubMed

大模型驱动的PubMed中文搜索引擎

马上搜索

文档翻译

学术文献翻译模型，支持多种主流文档格式。

立即体验