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Indium(III) chloride-catalyzed one-pot synthesis of dihydropyrimidinones by a three-component coupling of 1,3-dicarbonyl compounds, aldehydes, and urea: an improved procedure for the Biginelli reaction.

作者信息

Ranu B C, Hajra A, Jana U

机构信息

Department of Organic Chemistry, Indian Association for the Cultivation of Science, Jadavpur, Calcutta 700 032, India.

出版信息

J Org Chem. 2000 Sep 22;65(19):6270-2. doi: 10.1021/jo000711f.

DOI:10.1021/jo000711f
PMID:10987976
Abstract
摘要

相似文献

1
Indium(III) chloride-catalyzed one-pot synthesis of dihydropyrimidinones by a three-component coupling of 1,3-dicarbonyl compounds, aldehydes, and urea: an improved procedure for the Biginelli reaction.氯化铟（III）催化1,3 - 二羰基化合物、醛和尿素的三组分偶联一锅法合成二氢嘧啶酮：一种改进的Biginelli反应方法。
J Org Chem. 2000 Sep 22;65(19):6270-2. doi: 10.1021/jo000711f.
2
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Indium-catalyzed highly efficient three-component coupling of aldehyde, alkyne, and amine via C-H bond activation.铟催化的通过C-H键活化实现醛、炔烃和胺的高效三组分偶联反应。
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Copper nitrate catalyzed three-component one-pot synthesis of 3,4-dihydropyrimidin-2(1H)-ones.硝酸铜催化的3,4-二氢嘧啶-2(1H)-酮的三组分一锅法合成
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Demonstration of the feasibility of a direct solid-phase split-pool Biginelli synthesis of 3,4-dihydropyrimidinones.3,4-二氢嘧啶酮直接固相拆分池法Biginelli合成的可行性证明
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7
One-pot synthesis of 3,4-dihydropyrimidin-2(1H)-ones using chloroacetic acid as catalyst.以氯乙酸为催化剂一锅法合成3,4-二氢嘧啶-2(1H)-酮
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Indium-mediated asymmetric barbier-type allylations: additions to aldehydes and ketones and mechanistic investigation of the organoindium reagents.铟介导的不对称巴尔比耶型烯丙基化反应：醛和酮的加成反应及有机铟试剂的反应机理研究。
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Indium(III) chloride catalyzed three-component coupling reaction: a novel synthesis of 2-substituted aryl(indolyl)kojic acid derivatives as potent antifungal and antibacterial agents.三氯化铟催化的三组分偶联反应：新型 2-取代芳基（吲哚基）洛索酸衍生物的合成及其作为强效抗真菌和抗菌剂的研究。
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One-pot synthesis of 1,2,3-triazole linked dihydropyrimidinones via Huisgen 1,3-dipolar/Biginelli cycloaddition.一锅法合成 1,2,3-三唑并二氢嘧啶酮通过 Huisgen 1,3-偶极环加成/Biginelli 环加成。
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