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本文引用的文献

1
Nanocrystals: industrially feasible multifunctional formulation technology for poorly soluble actives.纳米晶体:难溶性活性药物工业可行的多功能制剂技术。
Int J Pharm. 2010 Oct 31;399(1-2):129-39. doi: 10.1016/j.ijpharm.2010.07.044. Epub 2010 Jul 30.
2
Preparation of hydrocortisone nanosuspension through a bottom-up nanoprecipitation technique using microfluidic reactors.使用微流控反应器通过自下而上的纳米沉淀技术制备氢化可的松纳米混悬液。
Int J Pharm. 2009 Jun 22;375(1-2):107-13. doi: 10.1016/j.ijpharm.2009.03.029. Epub 2009 Apr 5.
3
A novel bottom-up process to produce drug nanocrystals: controlled crystallization during freeze-drying.一种制备药物纳米晶体的新型自下而上方法:冷冻干燥过程中的控制结晶
J Control Release. 2008 Jun 4;128(2):179-83. doi: 10.1016/j.jconrel.2008.03.002. Epub 2008 Mar 7.
4
Nanosuspensions in drug delivery.药物递送中的纳米混悬液。
Nat Rev Drug Discov. 2004 Sep;3(9):785-96. doi: 10.1038/nrd1494.
5
Improvement of dissolution rates of poorly water soluble APIs using novel spray freezing into liquid technology.使用新型喷雾冷冻成液技术提高难溶性活性药物成分的溶出速率
Pharm Res. 2002 Sep;19(9):1278-84. doi: 10.1023/a:1020390422785.
6
Improving drug solubility for oral delivery using solid dispersions.使用固体分散体提高口服给药的药物溶解度。
Eur J Pharm Biopharm. 2000 Jul;50(1):47-60. doi: 10.1016/s0939-6411(00)00076-x.

Bottom-up preparation techniques for nanocrystals of lipophilic drugs.

作者信息

de Waard Hans, Frijlink Henderik W, Hinrichs Wouter L J

机构信息

Department of Pharmaceutical Technology and Biopharmacy, University of Groningen, Antonius Deusinglaan 1, 9713 AV Groningen, The Netherlands.

出版信息

Pharm Res. 2011 May;28(5):1220-3. doi: 10.1007/s11095-010-0323-3. Epub 2010 Nov 18.

DOI:10.1007/s11095-010-0323-3
PMID:21086152
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC3073053/
Abstract
摘要