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本文引用的文献

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A biomimetic synthesis of thiazolines using hexaphenyloxodiphosphonium trifluoromethanesulfonate.使用三氟甲磺酸六苯基氧代二鏻进行噻唑啉的仿生合成。
Angew Chem Int Ed Engl. 2003 Jan 3;42(1):83-5. doi: 10.1002/anie.200390059.
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ABC efflux pump-based resistance to chemotherapy drugs.基于ABC外排泵的化疗药物耐药性。
Chem Rev. 2009 Jul;109(7):2989-3011. doi: 10.1021/cr9000226.
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Structure of P-glycoprotein reveals a molecular basis for poly-specific drug binding.P-糖蛋白的结构揭示了多特异性药物结合的分子基础。
Science. 2009 Mar 27;323(5922):1718-22. doi: 10.1126/science.1168750.
4
Synthesis of libraries of thiazole, oxazole and imidazole-based cyclic peptides from azole-based amino acids. A new synthetic approach to bistratamides and didmolamides.由基于唑的氨基酸合成噻唑、恶唑和咪唑基环肽文库。一种合成双层酰胺和双莫拉酰胺的新方法。
Org Biomol Chem. 2007 May 21;5(10):1541-53. doi: 10.1039/b701999h. Epub 2007 Apr 16.
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Peptide-embedded heterocycles by mild single and multiple Aza-Wittig ring closures.通过温和的单步和多步氮杂维蒂希环化反应制备嵌入肽的杂环化合物。
Angew Chem Int Ed Engl. 2007;46(15):2701-3. doi: 10.1002/anie.200604507.
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Targeting multidrug resistance in cancer.针对癌症中的多药耐药性
Nat Rev Drug Discov. 2006 Mar;5(3):219-34. doi: 10.1038/nrd1984.
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Valspodar: current status and perspectives.
Expert Opin Investig Drugs. 1999 Jun;8(6):807-35. doi: 10.1517/13543784.8.6.807.
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Do drug substrates enter the common drug-binding pocket of P-glycoprotein through "gates"?药物底物是否通过“通道”进入P-糖蛋白的共同药物结合口袋?
Biochem Biophys Res Commun. 2005 Apr 8;329(2):419-22. doi: 10.1016/j.bbrc.2005.01.134.
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Thiopeptide antibiotics.硫肽类抗生素。
Chem Rev. 2005 Feb;105(2):685-714. doi: 10.1021/cr0300441.
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Simultaneous binding of two different drugs in the binding pocket of the human multidrug resistance P-glycoprotein.两种不同药物同时结合于人多药耐药性P-糖蛋白的结合口袋中。
J Biol Chem. 2003 Oct 10;278(41):39706-10. doi: 10.1074/jbc.M308559200. Epub 2003 Aug 7.

Design and synthesis of Selenazole-containing peptides for cocrystallization with P-glycoprotein.

作者信息

Tao Houchao, Weng Yue, Zhuo Rupeng, Chang Geoffrey, Urbatsch Ina L, Zhang Qinghai

机构信息

Department of Molecular Biology, The Scripps Research Institute, La Jolla, CA 92037, USA.

出版信息

Chembiochem. 2011 Apr 11;12(6):868-73. doi: 10.1002/cbic.201100048. Epub 2011 Mar 8.

DOI:10.1002/cbic.201100048
PMID:21387512
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC4814162/
Abstract
摘要