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通过N-连接的炔-烯醇立体和区域选择性合成4-乙烯基吡咯烷。

Stereo- and Regioselective Synthesis of 4-Vinylpyrrolidine from N-Tethered Alkyne-Alkenol.

作者信息

Devi Ngangbam Renubala, Behera Bipin K, Saikia Anil K

机构信息

Department of Chemistry, Indian Institute of Technology Guwahati, Guwahati 781039, India.

出版信息

ACS Omega. 2018 Jan 18;3(1):576-584. doi: 10.1021/acsomega.7b01785. eCollection 2018 Jan 31.

DOI:10.1021/acsomega.7b01785
PMID:31457915
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC6641446/
Abstract

Indium(III) chloride can be efficiently used for the synthesis of 4-vinylpyrrolidine from N-tethered alkyne-alkenol in good yields. The reaction is highly stereo- and regioselective.

摘要

氯化铟(III)可有效地用于由N-连接的炔-烯醇合成4-乙烯基吡咯烷，产率良好。该反应具有高度的立体选择性和区域选择性。

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本文引用的文献

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