咪唑啉的受体相互作用。I. 对大鼠主动脉α肾上腺素能受体的亲和力和效能。 - Suppr

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超能文献

Receptor interactions of imidazolines. I. Affinity and efficacy for alpha adrenergic receptors in rat aorta.

作者信息

Ruffolo R R, Rosing E L, Waddell J E

出版信息

J Pharmacol Exp Ther. 1979 Jun;209(3):429-36.

PMID:35606

Abstract

摘要

相似文献

Receptor interactions of imidazolines. I. Affinity and efficacy for alpha adrenergic receptors in rat aorta.咪唑啉的受体相互作用。I. 对大鼠主动脉α肾上腺素能受体的亲和力和效能。

J Pharmacol Exp Ther. 1979 Jun;209(3):429-36.

Receptor interactions of imidazolines. II. Affinities and efficacies of hydroxy-substituted tolazoline derivatives in rat aorta.咪唑啉的受体相互作用。II. 羟基取代妥拉唑啉衍生物在大鼠主动脉中的亲和力和效能。

J Pharmacol Exp Ther. 1979 Oct;211(1):74-9.

Receptor interactions of imidazolines. IV. Structural requirements for alpha adrenergic receptor occupation and receptor activation by clonidine and a series of structural analogs in rat aorta.咪唑啉的受体相互作用。IV. 可乐定及一系列结构类似物在大鼠主动脉中占据α肾上腺素能受体和激活受体的结构要求。

J Pharmacol Exp Ther. 1980 May;213(2):267-72.

Receptor interactions of imidazolines. III. Structure-activity relationships governing alpha adrenergic receptor occupation and receptor activation for mono- and dimethoxy-substituted tolazoline derivatives in rat aorta.咪唑啉的受体相互作用。III. 大鼠主动脉中一甲氧基和二甲氧基取代的妥拉唑啉衍生物对α肾上腺素能受体占据和受体激活的构效关系。

J Pharmacol Exp Ther. 1979 Dec;211(3):733-8.

[3H]Dihydroergocryptine binding to alpha adrenergic receptors in canine aortic membranes.[3H]双氢麦角隐亭与犬主动脉膜中α肾上腺素能受体的结合

J Pharmacol Exp Ther. 1978 Mar;204(3):606-14.

Aromatic and benzylic hydroxyl substitution of imidazolines and phenethylamines: differences in activity at alpha-1 and alpha-2 adrenergic receptors.咪唑啉和苯乙胺的芳族和苄基羟基取代：α-1和α-2肾上腺素能受体活性的差异。

J Pharmacol Exp Ther. 1983 Mar;224(3):559-66.

Receptor interactrions of imidazolines. VI. Significance of carbon bridge separating phenyl and imidazoline rings of tolazoline-like alpha adrenergic imidazolines.咪唑啉的受体相互作用。VI. 托拉唑啉样α肾上腺素能咪唑啉中分隔苯基和咪唑啉环的碳桥的意义。

J Pharmacol Exp Ther. 1980 Sep;214(3):535-40.

A comparison of pre- and postsynaptic alpha-adrenergic effects of phenylephrine and tramazoline on blood vessels of the rabbit in vivo.去氧肾上腺素和曲马唑啉对家兔体内血管的突触前和突触后α-肾上腺素能效应比较。

Naunyn Schmiedebergs Arch Pharmacol. 1978 Oct;304(3):223-30. doi: 10.1007/BF00507962.

Dissociation of alpha adrenergic receptor protection from inhibition of H-phenoxybenlamine binding in vascular tissue.α肾上腺素能受体保护作用与血管组织中H-酚苄明结合抑制的解离。

J Pharmacol Exp Ther. 1973 Jul;186(1):100-8.

On the capacity of presynaptic alpha receptors to modulate norepinephrine release from slices of rat neocortex and the affinity of some agonists and antagonists for these receptors.关于突触前α受体调节大鼠新皮质切片中去甲肾上腺素释放的能力以及一些激动剂和拮抗剂对这些受体的亲和力。

J Pharmacol Exp Ther. 1979 Dec;211(3):445-51.

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Agonist binding, agonist affinity and agonist efficacy at G protein-coupled receptors.G蛋白偶联受体的激动剂结合、激动剂亲和力和激动剂效能

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Receptor interactions of imidazolines: alpha-adrenoceptors of rat and rabbit aortae differentiated by relative potencies, affinities and efficacies of imidazoline agonists.咪唑啉的受体相互作用：通过咪唑啉激动剂的相对效价、亲和力和效能区分大鼠和兔主动脉的α-肾上腺素能受体

Br J Pharmacol. 1982 Sep;77(1):169-76. doi: 10.1111/j.1476-5381.1982.tb09283.x.

Analysis of the beta 1 and beta 2 adrenoceptor interactions of the partial agonist, clenbuterol (NAB365), in the rat jugular vein and atria.大鼠颈静脉和心房中部分激动剂克仑特罗（NAB365）的β1和β2肾上腺素能受体相互作用分析。

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Non-competitive antagonism of the alpha-adrenoceptor-mediated fast component of contraction of rat aorta, by doxazosin and prazosin.多沙唑嗪和哌唑嗪对大鼠主动脉α-肾上腺素能受体介导的快速收缩成分的非竞争性拮抗作用。

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