作为治疗阿尔茨海默病的天冬氨酸内肽酶（AEP）调节剂的3-炔基羧酰胺
3-Alkynyl Carboxamides as AEP Modulators for Treating Alzheimer's Disease.
作者信息
Sabnis Ram W, Sabnis Anika R
机构信息
Smith, Gambrell & Russell LLP, 1105 W. Peachtree Street NE, Suite 1000, Atlanta, Georgia 30309, United States.
Neuroscience Institute, Georgia State University, Atlanta, Georgia 30303, United States.
出版信息
ACS Med Chem Lett. 2024 Jan 4;15(2):159-160. doi: 10.1021/acsmedchemlett.3c00544. eCollection 2024 Feb 8.
Abstract
Provided herein are novel 3-alkynyl carboxamides as AEP modulators, their pharmaceutical compositions, the use of such compounds in treating Alzheimer's disease, and processes for preparing such compounds.
摘要
本文提供了作为AEP调节剂的新型3-炔基羧酰胺、它们的药物组合物、此类化合物在治疗阿尔茨海默病中的用途以及制备此类化合物的方法。
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本文引用的文献
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