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Remimazolam versus propofol for sedation in gastrointestinal endoscopy and colonoscopy within elderly patients: a meta-analysis of randomized controlled trials.老年患者胃肠内镜检查和结肠镜检查中瑞米唑仑与丙泊酚镇静效果的比较:一项随机对照试验的荟萃分析
Eur J Clin Pharmacol. 2024 Apr;80(4):493-503. doi: 10.1007/s00228-024-03624-6. Epub 2024 Jan 23.
2
Finding the ideal sedative: a non-inferiority study of remimazolam vs propofol in endoscopic retrograde cholangiopancreatography.寻找理想的镇静剂:瑞马唑仑与丙泊酚用于内镜逆行胰胆管造影术的非劣效性研究。
J Gastroenterol Hepatol. 2023 Dec;38(12):2160-2166. doi: 10.1111/jgh.16354. Epub 2023 Sep 20.
3
Remimazolam and serious adverse events: A scoping review.瑞马唑仑与严重不良事件:一项范围综述。
Eur J Anaesthesiol. 2023 Nov 1;40(11):841-853. doi: 10.1097/EJA.0000000000001902. Epub 2023 Sep 18.
4
Comparison of 95% effective dose of remimazolam besylate and propofol for gastroscopy sedation on older patients: A single-centre randomized controlled trial.甲磺酸瑞马唑仑与丙泊酚用于老年患者胃镜检查镇静的 95%有效剂量比较:一项单中心随机对照试验。
Br J Clin Pharmacol. 2023 Nov;89(11):3401-3410. doi: 10.1111/bcp.15839. Epub 2023 Jul 20.
5
Respiratory complications during recovery from gastrointestinal endoscopies performed by gastroenterologists under moderate sedation.胃肠病学家在适度镇静下进行胃肠内镜检查后恢复过程中的呼吸并发症。
Clin Endosc. 2023 Mar;56(2):188-193. doi: 10.5946/ce.2022.033. Epub 2023 Jan 10.
6
Effect of Remimazolam Tosilate on Respiratory Depression in Elderly Patients Undergoing Gastroscopy: A Multicentered, Prospective, and Randomized Study.甲苯磺酸瑞马唑仑对老年胃镜检查患者呼吸抑制的影响:一项多中心、前瞻性、随机研究。
Drug Des Devel Ther. 2022 Dec 5;16:4151-4159. doi: 10.2147/DDDT.S391147. eCollection 2022.
7
Remimazolam versus propofol for deep sedation/anaesthesia in upper gastrointestinal endoscopy in elderly patients: A multicenter, randomized controlled trial.瑞马唑仑与丙泊酚用于老年患者上消化道内镜检查中的深度镇静/麻醉:一项多中心、随机对照试验。
J Clin Pharm Ther. 2022 Dec;47(12):2230-2236. doi: 10.1111/jcpt.13797. Epub 2022 Nov 5.
8
New sedatives and analgesic drugs for gastrointestinal endoscopic procedures.用于胃肠内镜检查的新型镇静和镇痛药物。
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The hemodynamic stability of remimazolam compared with propofol in patients undergoing endoscopic submucosal dissection: A randomized trial.内镜黏膜下剥离术患者中瑞马唑仑与丙泊酚相比的血流动力学稳定性:一项随机试验。
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2021 Korean Society of Gastrointestinal Endoscopy Clinical Practice Guidelines for Endoscopic Sedation.2021年韩国胃肠内镜学会内镜镇静临床实践指南
Clin Endosc. 2022 Mar;55(2):167-182. doi: 10.5946/ce.2021.282. Epub 2022 Feb 22.

瑞马唑仑,一种新型药物,用于安全有效的内镜镇静。

Remimazolam, a novel drug, for safe and effective endoscopic sedation.

作者信息

Lee Jae Min, Park Yehyun, Ahn Dong Won, Lee Jun Kyu, Lee Kwang Hyuck

机构信息

Department of Internal Medicine, Korea University Anam Hospital, Seoul, Korea.

Department of Internal Medicine, Ewha Womans University Seoul Hospital, Seoul, Korea.

出版信息

Clin Endosc. 2025 May;58(3):370-376. doi: 10.5946/ce.2024.026. Epub 2025 Jan 14.

DOI:10.5946/ce.2024.026
PMID:39806820
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC12138356/
Abstract

Remimazolam is a novel benzodiazepine with unique pharmacokinetic and pharmacodynamic properties, making it an ideal candidate for sedation during endoscopic procedures. Distinguished by its rapid onset and short duration of action, remimazolam offers a safer and more efficient alternative to traditional sedatives, such as midazolam and propofol, with fewer side effects, such as hypotension, bradycardia, and respiratory depression. This article reviews the characteristics of remimazolam and its practical advantages, including ease of use, quick recovery time, and minimal residual sedation, emphasizing its potential to improve patient safety and procedural efficiency in clinical endoscopy settings.

摘要

瑞马唑仑是一种新型苯二氮䓬类药物,具有独特的药代动力学和药效学特性,使其成为内镜手术镇静的理想选择。瑞马唑仑以其起效迅速和作用时间短为特点,与咪达唑仑和丙泊酚等传统镇静剂相比,提供了一种更安全、更有效的替代方案,副作用更少,如低血压、心动过缓和呼吸抑制。本文综述了瑞马唑仑的特点及其实际优势,包括使用方便、恢复时间快和残余镇静作用极小,强调了其在临床内镜检查中提高患者安全性和手术效率的潜力。