去甘氨酰胺9-赖氨酸加压素对吗啡镇痛耐受性形成的促进作用。
Facilitation of development of resistance to morphine analgesia by desglycinamide9-lysine vasopressin.
作者信息
Krivoy W A, Zimmermann E, Lande S
出版信息
Proc Natl Acad Sci U S A. 1974 May;71(5):1852-6. doi: 10.1073/pnas.71.5.1852.
Abstract
Desglycinamide(9)-lysine vasopressin facilitates development of resistance to the analgesic action of morphine in mice if morphine is administered before the peptide. Desglycinamide(9)-lysine vasopressin is not a morphine antagonist, and does not appear to cause either hyperalgesia or alteration of the response to the technique used for evaluating analgesia.
摘要
如果在给予去甘氨酰胺（9）-赖氨酸加压素之前给予吗啡，去甘氨酰胺（9）-赖氨酸加压素会促进小鼠对吗啡镇痛作用产生耐受性。去甘氨酰胺（9）-赖氨酸加压素不是吗啡拮抗剂，似乎既不会引起痛觉过敏，也不会改变用于评估镇痛的技术所产生的反应。
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