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Synthesis of 6-phenanthridinones and their heterocyclic analogues through palladium-catalyzed sequential aryl-aryl and N-aryl coupling.

作者信息

Ferraccioli Raffaella, Carenzi Davide, Rombolà Ottavio, Catellani Marta

机构信息

CNR-Istituto di Scienze e Tecnologie Molecolari (ISTM), Dipartimento di Chimica Organica e Industriale, Università di Milano, Via C. Golgi 19, 20133 Milano, Italy.

出版信息

Org Lett. 2004 Dec 9;6(25):4759-62. doi: 10.1021/ol0479949.

DOI:10.1021/ol0479949
PMID:15575679
Abstract

[reaction: see text] 6-Phenanthridinones and their heterocyclic analogues were synthesized through a one-pot procedure based on consecutive Pd-catalyzed aryl-aryl and N-aryl coupling from iodoarenes ortho-substituted by electron-releasing substituents and amides of o-bromoarene- and heteroarenecarboxylic acids.

摘要

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