Trichloromethylthiolation of N-Heterocycles: Practical and Completely Regioselective.
作者信息
Ernst Johannes B, Rühling Andreas, Wibbeling Birgit, Glorius Frank
机构信息
Organisch-Chemisches Institut, Westfälische Wilhelms-Universität Münster, Corrensstraße 40, 48149, Münster, Germany.
出版信息
Chemistry. 2016 Mar 18;22(13):4400-4. doi: 10.1002/chem.201600377. Epub 2016 Feb 16.
PMID:26833581
Abstract
The first trichloromethylthiolation of a broad range of indoles and pyrroles is reported employing bench-stable N-trichloromethylthiosaccharin as reagent. This methodology is highly regioselective, exhibits high functional group tolerance, and provides access to two previously unknown classes of potentially bioactive compounds.
摘要
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