2-氨基苯并咪唑酰胺衍生物的合成、抗血脂及血小板抗聚集活性
Synthesis, antilipidemic and platelet antiaggregatory activity of 2-aminobenzimidazole amide derivatives.
作者信息
Caroti P, Ceccotti C, Da Settimo F, Primofiore G, Franzone J S, Reboani M C, Cravanzola C
机构信息
Istituto di Chimica Farmaceutica, Università di Pisa, Italy.
出版信息
Farmaco. 1989 Mar;44(3):227-55.
PMID:2775417
Abstract
The synthesis and preliminary pharmacological evaluation of 2-aminobenzimidazole amide derivatives are reported. None of these compounds showed antilipidemic or platelet antiaggregatory activity comparable to that of drugs used in therapy.
摘要
报道了2-氨基苯并咪唑酰胺衍生物的合成及初步药理评价。这些化合物均未表现出与治疗中使用的药物相当的抗血脂或血小板抗聚集活性。
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