Chen Jing-Biao, Jia Yi-Xia
College of Chemical Engineering, Zhejiang University of Technology, Hangzhou 310014, China.
Org Biomol Chem. 2017 May 3;15(17):3550-3567. doi: 10.1039/c7ob00413c.
Numerous efficient synthetic methods for enantioselective indole functionalizations have emerged in recent years. This review summarizes the major achievements in the transition-metal-catalyzed enantioselective indole functionalization reactions since 2010 and focuses on C-C bond formation processes, including alkylations, arylations, cycloaddition reactions, and other reactions. It intends to give a compendious overview of the significant progress achieved in this area.
近年来,出现了许多用于对映选择性吲哚官能团化的高效合成方法。本综述总结了自2010年以来过渡金属催化的对映选择性吲哚官能团化反应的主要成就,并重点关注C-C键形成过程,包括烷基化、芳基化、环加成反应及其他反应。其旨在对该领域取得的重大进展进行简要概述。