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本文引用的文献

1
DETERMINATION OF A PROTONATION SCHEME OF TETRACYCLINE USING NUCLEAR MAGNETIC RESONANCE.
Anal Chem. 1965 Jun;37:872-5. doi: 10.1021/ac60226a022.
2
Avidity of the tetracyclines for the cations of metals.四环素对金属阳离子的亲合力。
Nature. 1956 Mar 3;177(4505):433-4. doi: 10.1038/177433a0.
3
Active efflux of tetracycline encoded by four genetically different tetracycline resistance determinants in Escherichia coli.大肠杆菌中由四种基因不同的四环素抗性决定簇编码的四环素主动外排
Proc Natl Acad Sci U S A. 1980 Jul;77(7):3974-7. doi: 10.1073/pnas.77.7.3974.
4
Transport of the lipophilic analog minocycline differs from that of tetracycline in susceptible and resistant Escherichia coli strains.在敏感和耐药的大肠杆菌菌株中，亲脂性类似物米诺环素的转运与四环素不同。
Antimicrob Agents Chemother. 1982 Nov;22(5):791-9. doi: 10.1128/AAC.22.5.791.
5
Tetracycline diffusion through phospholipid bilayers and binding to phospholipids.四环素通过磷脂双分子层的扩散及其与磷脂的结合。
Antimicrob Agents Chemother. 1984 Aug;26(2):263-5. doi: 10.1128/AAC.26.2.263.
6
Tetracyclines of various hydrophobicities as a probe for permeability of Escherichia coli outer membranes.不同疏水性四环素作为大肠杆菌外膜通透性的探针
Antimicrob Agents Chemother. 1984 May;25(5):539-44. doi: 10.1128/AAC.25.5.539.
7
Energetics of tetracycline transport into Escherichia coli.四环素转运至大肠杆菌的能量学
Antimicrob Agents Chemother. 1984 Apr;25(4):446-9. doi: 10.1128/AAC.25.4.446.
8
Stoichiometry of the H+-ATPase of growing and resting, aerobic Escherichia coli.生长和静止的好氧大肠杆菌H⁺-ATP酶的化学计量学
Biochemistry. 1982 Oct 26;21(22):5534-8. doi: 10.1021/bi00265a024.
9
Antibiotic uptake by bacteria as measured by partition in polymer aqueous phase systems.通过聚合物水相体系中的分配来测定细菌对抗生素的摄取。
Anal Biochem. 1984 Aug 15;141(1):94-100. doi: 10.1016/0003-2697(84)90430-5.
10
Permeability of lipid bilayer membranes to organic solutes.脂质双分子层膜对有机溶质的通透性。
J Gen Physiol. 1968 Sep;52(3):495-508. doi: 10.1085/jgp.52.3.495.

Penetration of lipophilic agents with multiple protonation sites into bacterial cells: tetracyclines and fluoroquinolones as examples.

作者信息

Nikaido H, Thanassi D G

机构信息

Department of Molecular and Cell Biology, University of California, Berkeley 94720.

出版信息

Antimicrob Agents Chemother. 1993 Jul;37(7):1393-9. doi: 10.1128/AAC.37.7.1393.

DOI:10.1128/AAC.37.7.1393
PMID:8363364
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC187981/
Abstract
摘要