Department of Chemistry, University of Pennsylvania, Philadelphia, Pennsylvania 19104-6323, USA.
Org Lett. 2011 Mar 4;13(5):1242-5. doi: 10.1021/ol200128y. Epub 2011 Feb 4.
A large array of aryl and heteroaryl mesylates have been successfully employed as electrophiles in a Csp(2)-Csp(3) Suzuki-Miyaura cross-coupling with potassium ammonio- and amidomethyltrifluoroborates to afford the corresponding products in high yields.
大量芳基和杂芳基甲磺酸酯已成功用作亲电试剂,与氨甲基金和氨甲基三氟硼酸钾进行 Csp(2)-Csp(3)Suzuki-Miyaura 交叉偶联,以高产率得到相应的产物。