State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Gansu Lanzhou, 730000, PR China.
J Org Chem. 2013 Mar 15;78(6):2746-50. doi: 10.1021/jo302555z. Epub 2013 Feb 21.
A simple route for the synthesis of imidazole derivatives via copper-catalyzed [3 + 2] cycloaddition reaction is described. This strategy has achieved high regioselectivity and used oxygen as an oxidant without the addition of expensive catalysts to provide moderate to good yields.
本文描述了一种通过铜催化的[3 + 2]环加成反应合成咪唑衍生物的简单路线。该策略具有高区域选择性，并使用氧气作为氧化剂，无需添加昂贵的催化剂，即可提供中等至良好的产率。
