Birman Vladimir B, Li Ximin
Department of Chemistry, Washington University, Campus Box 1134, One Brookings Drive, St. Louis, Missouri 63130, USA.
Org Lett. 2006 Mar 30;8(7):1351-4. doi: 10.1021/ol060065s.
[reaction: see text] A commercially available pharmaceutical, tetramisole, was found to be a competent enantioselective acylation catalyst. Its benzannellated analogue, benzotetramisole (BTM), produced outstanding enantioselectivities in kinetic resolution of secondary benzylic alcohols.
[反应：见正文] 一种市售药物四咪唑被发现是一种有效的对映选择性酰化催化剂。其稠合苯类似物苯并四咪唑（BTM）在仲苄醇的动力学拆分中产生了出色的对映选择性。
