Key Laboratory of Natural Medicine and Immuno-Engineering of Henan Province, Henan University, Jinming Campus, Kaifeng, Henan 475004, China PR.
Org Lett. 2010 May 21;12(10):2234-7. doi: 10.1021/ol100586r.
A rapid and efficient synthesis of 2H-indazoles has been developed, which involves the [3 + 2] dipolar cycloaddition of arynes and sydnones. The process proceeds under mild reaction conditions in good to excellent yields.
一种快速高效的 2H-吲唑合成方法已经被开发出来,该方法涉及芳炔和 sydnones 的 [3 + 2] 偶极环加成反应。该过程在温和的反应条件下以良好到优异的收率进行。